"目錄號: HY-13724B

Others-

Pipendoxifene hydrochloride 是一種選擇性的雌激素受體調(diào)節(jié)劑 (SERMs)。

Estrogen Receptor/ERR

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生物活性

Description

Pipendoxifene hydrochloride is a selectiveestrogen receptormodulators (SERMs).

IC50& Target

Estrogen receptor[1]

In Vitro

Pipendoxifene is a new 2-phenyl indole selective estrogen receptor modulators (SERM) that exhibits an excellent preclinical pharmacological profile and is selected for further development as a treatment for metastatic breast cancer[1].

References

[1].Shelly W,? et al. Selective estrogen receptor modulators: an update on recent clinical findings. Obstet Gynecol Surv. 2008 Mar;63(3):163-81.